Mero ea litholoana tsa morara e thibela ho senyeha ha meriana e meng.
Ha e le hantle, lero la morara le qhibilihisitsoeng ke li-vithamine le limatlafatsi. Bakeng sa ba bangata, khalase ea lero la morara ke tsela e nepahetseng ea ho qala letsatsi. Leha ho le joalo, haeba u na le meriana e itseng, e kang meriana e itseng ea pelo e bitsoang statins, u lokela ho qoba ho noa lero la morara ha u noa meriana ena. Jero ea litholoana tsa morara e ka thibela 'mele oa hao ho khona ho senya meriana ena, e leng eona e ka lebisang liphellong tse bohloko.
Mero ea litholoana tsa morara le Statements e itseng U se ke Ua Kopanya
Sejo sa litholoana tsa morara le li-statins tse itseng (tse sebelisoang ho phekola k'holeseterole e phahameng) tse kang Lipitor (atorvastatin), Mevacor (lovastatin), le Zocor (simvastatin) ha li kopane. Sejo sa litholoana tsa morara se sitisa mokhoa oa li-enzyme tse thusang ho senya meriana e ngata, ho akarelletsa Lipitor, Mevacor le Zocor .
Haeba u noa lero la morara ha u ntse u noa meriana leha e le efe, lithethefatsi tse ngata haholo li ka kena ka mali a hao. Sena se ka baka liphello tse bohloko, tse kang ho kula ha mesifa kapa kotsi ea sebete. Ka ho khetheha, lero la morara le thibela lipilisi tsa enzyme ea hepatic (sebete) P450, e senyang lithethefatsi.
Ka ho senya le enzyme ea sebete, motsoako o sebetsang haholo o ama 'mele oa hau. Ka mantsoe a mang, liphello tsa lithethefatsi tsa statin li eketseha ho batho ba noang lero la lamunu. Litholoana tse mpe tsa li-statins li kenyeletsa tšenyo ea mesifa le sebete.
Li-enzyme tsa Cytochrome P450 li bolokiloe li-cell reticulum tse se fumaneng feela sebeteng empa hape le liphio, pampiri ea meno le matšoafo.
Li-enzyme tsena tsa P450 li senya lithethefatsi fatše ka ho li fa oxidizing. Ho phaella ho lero la litholoana tsa morara, ho na le lintho tse ling tse thibelang li-enzyme tsa cytochrome P450 tse nang le li-enzyme tse kang cimetidine (histamine blocker e sebelisetsoang ho phekola GERD), erythromycin (lithibela-mafu) le isoniazid (meriana e sebelisoang ho phekola lefuba).
Ke kopa u hopole hore ho na le lithethefatsi tse 'maloa tse senyang ka cytochrome P450,' me haeba u na le lipotso mabapi le likamano tse ka khonehang, ka kōpo buisana le ngaka ea hau. Ngaka ea hau e boetse e lokela ho hlahloba hore na meriana eo ue nkang e na le likamano tse se nang molekane kapa lijo tsa hau.
Nako eo u noang meriana ena ka eona le nako eo u jang litholoana tsa morara kapa ea noa lero la morara ha e fokotsa kotsi ea lits'ebeletso tse kotsi tse amanang le lithethefatsi - ho buisana ho ka etsahala ho fihlela matsatsi a mararo ka mor'a ho ja litholoana tsa morara. Sena se bolela hore o ke ke oa noa lero la litholoana tsa morara hoseng 'me u noa meriana ea hau hamorao motšehare.
Mekhoa ea Meriana
O na le likhetho tse 'maloa:
- U ka kenyelletsa litholoana tsa morara ho tsoa lijong tsa hau 'me u kenyelletsa litholoana tse ling le litholoana tsa litholoana, kapa
- Haeba u batla ho tsoela pele ho ja lihlahisoa tsa morara, bua le ngaka ea hau ka ho sebelisa meriana e meng.
Litšoantšo tse 'maloa tse fumanehang ha li sebelisane le lero la morara' me li sireletsehile ho li sebelisa. Tsena li kenyelletsa:
- Crestor (rosuvastatin)
- Lescol (fluvastatin)
- Pravachol (pravastatin)
Boitsebiso bo eketsehileng
Haeba u na le lipotso mabapi le ho sebelisana ha lithethefatsi le lero la morara, ka kōpo buisana le ngaka ea hau ka lintho tsena.
Ka kopo hopola hore ngaka ea hau ke mohloli o motle oa tlhahisoleseding mme o teng ho o thusa ho o tataisa kalafo mme o sebetse ho netefatsa bophelo ba hao bo botle.
Mehloli e khethiloeng
Article e nang le sehlooho se reng "Litšebelisano le lithethefatsi ka lebaka la cytochrome P450" ke CC Ogu le JL Maxa e hatisitsoeng Baylor University Medical Center Proceedings ka 2000.
Trevor AJ, Katzung BG, Kruidering-Hall M. Antifungal Agents. Ka: Trevor AJ, Katzung BG, Kruidering-Hall M. eds. Katzung & Trevor's Pharmacology: Ho hlahlojoa le ho hlahloba boto, 11e . New York, NY: Hill ea McGraw; 2015. Fihletsoe ka la 29 February, 2016.