Methimazole, Carbimazole le Propylthiouracil / PTU
Ha qoqotho ea qoqotho e fetoha ho feteletseng - boemo bo tsejoang e le hyperthyroidism - lesela le hlahisa hormone e ngata ea qoqotho. Sena se ka baka matšoao a sa tšoaneng, ho kopanyelletsa le ho phalla ka potlako, khatello e phahameng ea mali, ho tšoenyeha, ho hlobaela, ho thothomela, ho lahleheloa ke mali, letšollo, le matšoao a mangata a metabolism e feteletseng, le litšoelesa tse feteletseng le litho tsa 'mele.
Phekolo e kholo ea hyperthyroidism ke karolo ea meriana ea ngaka e tsejoang e le lithethefatsi tsa antithyroid. Lithethefatsi tsa Antithyroid li boetse li bitsoa li-thioamide. Ke lithethefatsi tse sebelisetsoang ho phekola thyroid e feteletseng - hyperthyroidism - ho kenyeletsa ha qoqotho e se e feteletse haholo ka lebaka la lefu la Graves, goiter tse ngata tse chefo, kapa li-nodules tse chefo.
Lithethefatsi tsa Antithyroid li sebetsa ka ho thibela bokhoni ba qoqotho ea bokhoni ba ho hlahisa lihomone tse peli tsa qoqotho thyroxine (T4) le triiodothyronine (T3).
Meriana e ka sehloohong ea li- antithroid e United States e fumaneha methimazole le propylthiouracil (PTU). Ka ntle ho United States, likhetho ke methimazole, carbimazole, le PTU.
Methimazole
Methimazole ea lithethefatsi ea antithyroid e thibela thyroid ho sebelisa iodine - hangata ho tsoa lijong kapa li-supplement - ho hlahisa hormone ea qoqotho. Ke meriana e atisang ho nkoa hang ka letsatsi ke bakuli.
Ka linako tse ling lebitso la maethimazole le bitsoa thiamazole.
Meriana ena e sebelisoa ho pota lefatše mme ke lithethefatsi tse ka sehloohong tsa li-antithyroid tse sebelisoang United States, moo e fumanehang tlasa lebitso la Tapazole.
Baetsi ba 'maloa ba boetse ba fana ka mofuta o tloaelehileng oa methimazole.
Carbimazole
Carbimazole ke sethethefatsi seo, ha se laoloa, se fetohela meriana ea methimazole 'meleng,' me ka hona se tšoana hantle le liketso.
Lejoe le tummeng ka ho fetisisa la carbimazole ke Neomercazole.
Neomercazole ke lebitso la carbimazole 'me le etsoa ke Amdipharm International (UK). Meriana eo e ne e lumelloa ka 2004, 'me e rekisoa UK le Europe, empa ha e fumanehe kapa e fanoe United States. U ka bona datasheet ho Neomercazole mona. Mona ke lisebelisoa tse 'maloa tse eketsehileng mabapi le Neomercazole.
- Websaete ea Moetsi oa Lithethefatsi: Amdipharm
- Ho hlalosa litaba
Neomercazole Lisebelisoa : carbimazole Ph.Eur; lactose; starch ea poone; sucrose; stearate ea magnesium; sucrose; talc; gum lemon; ferric oxide; propyl hydroxybenzoate; le gelatin.
Matla a fumanehang : 5 mg
Mabitso a mang / Mabitso: Carbimazole e fumaneha linaheng tse ling tsa Europe le Asia ka tlas'a mabitso a latelang: Atirozidina, Basolest, CG1, Carbimazole Spofa, Carbotiroid, Mertiran, Neo-Mercazole, Neo-Thyreostat, Neo-Tireol le Tyrazol.
Propylthiouracil / PTU
Tsela eo PTU e etsang hore qoqotho e fetotsoe ka eona ea qoqotho ea qoqotho ke hore e thibela qoqotho ea qoqotho ho sebelisa li-iodine ho hlahisa hormone ea qoqotho. E boetse e thibela phetoho ea hormone ea thyroid T4 ka T3. PTU e na le nako e khutšoanyane ea liketso, kahoo bakuli ba noang meriana ena hangata ba laeloa hore ba noe meriana ka makhetlo a mabeli ho isa ho a mararo ka letsatsi ho fokotsa li-hormone tsa qoqotho.
PTU e na le litla-morao tse ngata ho feta lithethefatsi tse ling tseo ho buuoang ka tsona mona, 'me ke moriana o khethiloeng bakeng sa hyperthyroidism feela maemong a' maloa (nakong ea bokhachane pele ho nako, sefefo se matla sa qoqotho le ha mokuli a e-ba le litla-morao tse tebileng tsa methimazole).
United States, PTU feela e fumaneha; ha ho na mabitso a maru a PTU a rekisoang United States. Bahlahisi ba bangata ba hlahisa PTU e tloaelehileng.
Boitsebiso bo eketsehileng
Ithute ho eketsehileng ka hyperthyroidism le mekhoa ea eona ea phekolo, ho akarelletsa le lithethefatsi tsa antithyroid, ho lisebelisoa tsena:
- Hyperthyroidism | 'Maloetse a Mabitla | Thyroid e feteletseng
- 'Maloetse a Mabitla le Hyperthyroidism 101
- Hyperthyroidism Likotsi / Matšoao a Palo
- Likotsi Tsa Mafu a Mabitla le Hyperthyroidism
- Lipotso Tse Atisang ho Botsoa Libukeng tsa Hyperthyroidism le Graves
- Litsela Tse 3 tsa ho Phekola Hyperthyroidism
Lisebelisoa:
Letsatsi le leng le le leng, Medina ea Lijo tsa Meriana ea Lijo le Lithethefatsi tsa US, Online
Tlhaloso ea Tšireletso ea Meriana ea FDA ea Meriana: Temoso e Ncha ea Lehloeo ka kotsi e matla ea sebete le propylthiouracil, la 21 April, 2010
Ross, Douglas MD, "Tlhaloso ea mokuli: Lithethefatsi tsa Antithyroid," UpToDate . Qetellong ea ntlafatsoa: la 13 November, 2009