Li-Triptans li lokisa li-migraine joang le seo u ka se hlokomelang
U ka 'na ua nka triptan-esita le ho e jara ka har'a mokotla oa hau kapa mokotlana oa chelete-ho fokotsa tlhaselo ea migraine hang ha e itlhahisa. Le hoja li-triptan li sireletsehile ebile li mamelloa hantle, ha li lumelle motho e mong le e mong.
Ho sebelisa Triptan bakeng sa Thuso ea Migraine
Li-triptans li sebelisetsoa ho tšoara migraine e itekanetseng le e matla, hammoho le migraine e bonolo e sa amoheleng meriana e fetang-ea-counter, joaloka antisteroidal anti-inflammatories .
Li ka boela tsa sebelisoa ho tšoara migraine e bonolo ho ea ho batho ba sa khoneng ho mamella kapa ho nka li-NSAID.
The Science Behind Triptans
Triptans li tlama ho li-receipton serotonin bokong. Ka ho etsa li-receptor serotonin, methapo ea mali bokong e fokolisitsoe 'me litsela tse ling tsa bokong bo koetsoe. Hape ho lumeloa hore Triptans e sebetsa ka ho fokotsa litekanyetso tsa CGRP -a protheine e phahame nakong ea tlhaselo ea migraine.
Mefuta e sa Tšoaneng
Triptans li ipiletsa hobane ho na le litsela tse fapa-fapaneng tseo ba ka li nkang. Ka mohlala, li-triptan li ka nkoa ka molomo, ka nko, esita le ho kenngoa ka nale ho lihlahisoa tse nonneng tsa motho (tse bitsoang sejoe sa subcutaneous). Hape ho na le triptan e bitsoang Maxalt XLT (rizatriptan) e ka qhalang ka potlako molomong oa motho 'me e kenngoa esita leha motho a hlatsa. Qetellong, Imitrex (sumatriptan) e ka fanoa e le letlotlo.
Phetoho e kholo hape ke letlalo la letlalo la triptan.
Zecuity (sumatriptan) ke patch transdermal patch e sebelisoang ke betri e tsamaisang sumatriptan ka letlalo la motho. Zecuity, hammoho le triptan e nang le injection, e ipiletsa ka ho khetheha bakeng sa ba nang le ho nyefoloha le ho hlatsa ba amanang le migraine ea bona. Ho boleloa hore, ka June 2016, FDA e ile ea nka Zecuity ho tsoa 'marakeng ka lebaka la mathata a ho chesa le maqeba a maholo ho batho ba sebelisang thepa.
Phuputso e ntse e tsoela pele.
Liketsahalo tse ka 'nang tsa e-ba teng
Triptans ke meriana e sebetsang ea migraine. Seo se boleloa, ke meriana ea meriana ebile e hloka ho nkoa tlas'a tlhokomelo ea ngaka. Tse ling tsa litla-morao tse tloaelehileng tse nang le triptans li kenyeletsa
- Nausea
- Tšoaea, molala, kapa sefubelu sa sefuba kapa khatello kapa maikutlo a ho hatella
- Lebelo la pelo kapele kapa le eketsa khatello ea mali
- Mokhathala
- Ho utloahala / ho utloa bohloko (haholo-holo sefahlehong)
- Ho utloahala ho utloahala ha letlalo
Triptans Ha e Bohle
Ke habohlokoa ho hlahloba nalane ea hau ea bongaka le meriana eohle ea hau, ho kenyeletsa li-supplement le li-vithamine tse ngata, le ngaka ea hau ea botho. Batho ba bang ha baa lokela ho nka triptan hobane ba ka mpefatsa maemo a bophelo bo botle. Ka mohlala, ha ua lokela ho nka triptan haeba u e-na le histori ea lefu la methapo ea 'mele , lefu la seoa , methapo ea lefuba , khatello ea mali e sa laoleheng, kapa hemiplegic kapa buslar migraine.
Li-triptans li boetse li hanyetsanoa le batho ba sebelisang monoamine oxidase inhibitors ka nako e le 'ngoe' me ha baa lokela ho sebelisoa ka letsatsi le le leng joaloka ergotamine kapa dihydroergotamine.
Hape, ho kopanya li-triptans tse khethiloeng-serotonin reuptake inhibitors (SSRIs) kapa khetho ea norepinephrine reuptake inhibitors (SNRIs) e ka fella ka lefu la serotonin.
Sena se ka 'na sa bolaea, le hoja se sa tloaeleha se ka bakang matšoao a sa tšoaneng a kang:
- pherekano
- pherekano
- letšollo
- ho fufuleloa
- ho felloa ke tekano
- ho thothomela
- ho thothomela
- feberu
Triptans lilemong tsa basali ba ho bela
Mabapi le bokhachane, triptan ke setho sa mofuta oa C, e leng se bolelang hore karolelano ea kotsi le molemo e lokela ho behoa ke ngaka bakeng sa mokuli ka mong. Mabapi le ho anyesa, dintlha tsa saense tsa ho sebelisa triptans bakeng sa phekolo ea migraine e lekanyelitsoe-le hoja, sumatriptan e nkoa e lumellana le American Academy of Pediatrics.
Haeba o nka triptan le moralo oa ho ima kapa ho anyesa, ka kopo bua le ngaka ea hau ho fumana moralo o molemo ka ho fetisisa oa phekolo.
Lentsoe le Tsoang ho
Litaba tse monate tsa li-triptan ke hore ho na le mefuta e mecha ea ho fana ka nako e ntseng e hlahisoa, e kang sesebelisi sa lipuo tsa sumatriptan, omitriptan inhaler le molomo oa rizatriptan ho qhala filimi.
Triptans ke mekhoa e metle ea ho phekola migraine ha e fanoa tlas'a tlhokomelo ea ngaka. Tsela e ikhethang ea tsamaiso e thusa haholo ka ho phekola ba nang le bothata ba ho nyefoloa le ho hlatsa ho amanang le migraine. E-ba moemeli oa bophelo ba hao ba migraine 'me u bue le ngaka ea hao ka hore na triptan e na le khetho e ntle ho uena.
Lisebelisoa:
Ables, A le Nagpilli R.Prevention, Tlhahlobo le Tsamaiso ea Serotonin Syndrome. Ke Mooki oa Lefu. 2010 Mantaha 1; 81 (9): 1139-1142.
Gilmore B, Michael M. Phekolo ea Bohlokoa ba Hlooho ea Migraine. Ke Mooki oa Lefu . 2011 Feb 1; 83 (3): 271-280.
Goldstein J, Smith TR, Pugach N, Griesser J, Sebree T, Pierce M. Sethatriptan iontophoretic transdermal tsamaiso ea phekolo e matla ea migraine. Hlooho ea hlooho . 2012 Oct; 52 (9): 1402-10.
Hutchinson S, Marmura MJ, Calhoun A, Lucas S, Silberstein S, Peterlin BL. Tšebeliso ea Litlhare tse Tloaelehileng tsa Migraine ho Basali ba Fepa Mabese: Kakaretso ea Litlhahiso. Hlooho ea hlooho. 2013 Mar; 53 (4): 614-27.
US Administration of Drug and Drug Administration. (6/2/2016). Zakuity (sumatriptan) Migraine Patch: Puisano ea tšireletso ea lithethefatsi - FDA kotsi ea ho hlahloba kotsi le maqeba.