Prezcobix (darunavir + cobicistat) ke motsoako o tsitsitseng o sebelisang phekolo ea HIV . Likarolo tse peli tsa lithethefatsi tse nang le Prezcobix li atisa ho rekisoa ho Prezista (darunavir) le Tybost (cobicistat) .
Pilisi e le 'ngoe, sebōpeho se entsoeng ka' ngoe e fana ka mokhoa o bonolo, hang-o mong le o mong, 'me motsoako oa li-cobicistat o matlafatsa le ho o boloka ka mahlaseli a plasma a Prezista' meleng.
Prezcobix e ile ea amoheloa ke US Food and Drug Administration (FDA) ka January 2015 bakeng sa bakuli ba bacha ba bacha le ba nang le phihlelo ba nang le tšoaetso ea HIV-1.
Foromo
Letlapa le koahetsoeng ka filimi le koahetsoeng ka filimi, le nang le 800mg la darunavir le 150mg la cobicistat, ke le pinki le 'mala o nang le "TG" ka lehlakore le le leng "800" ka lehlakoreng le leng.
Tekanyo
Letlapa le le leng le nkiloe letsatsi ka leng le lijo. Prezcobix e ke ke ea sebelisoa e le mong empa e lokela ho nkoa e kopane le e le 'ngoe kapa tse ling tse fapaneng le li-antiretroviral.
Litaelo
Pele ho qala, bakuli ba lokela ho hlahlojoa hore ba hlahlobe tumello ea bona ea tlhaho ea li-creatinine kaha Prezcobix e ka 'na ea baka tšenyo ea liphio, hangata ho bakuli ba nang le bothata ba ho se sebetse ba leihlo kapa ba sa tsejoeng. Ha e laoloa ke Viread (tenofovir) - moriana o tsejoang hape hore o bakile tšenyo ea likokoana-hloko hoa khothalletsoa hore bakuli ba hlahlojoe sekoloto sa tekanyetso ea creinine, glucose ea urese le protheine ea moroto.
Ho boetse ho kgothaletswa hore bakuli ba nang le phihlelo, haholo-holo ba pepesehileng ho HIV protease inhibitors , ba fanoe ka tlhahlobo ea liphatsa tsa lefutso pele ba nka Prezcobix. Haeba tlhahlobo ea genotypic e sa fumanehe, Prezcobix e lokela ho qojoa ho mang kapa mang ea neng a pepesehetse HIV protease inhibitors.
Liphello tse Tloaelehileng
Lipatlisisong tsa bongaka tsa Thuto ea bo-III, ho na le liphello tse ngata tsa lithethefatsi tse ka fumanoang ha u sebelisa Prezcobix. Liketsahalo tse bohloko ka ho fetisisa, tse tlalehiloeng ka 5% kapa tlase ho bakuli, e ne e le:
- Letšollo
- Nausea
- Rash
- Hlooho ea hlooho
- Mahlaba a mpa
- Ho otla
Litlhaloso tsa lithethefatsi
Prezcobix ha ea lokela ho nkoa ka lithethefatsi tse latelang kapa litlama tse tlatsetsang:
- Meriana e thibelang li-anginal: Ranexa
- Meriana e thibelang ho itšireletsa: Multaq
- Meriana ea anti-k'holeseterole: Mevacor, Zocor
- Meriana ea anti-gout: Uroxatral
- Meriana ea ho hatella meriana ea mali: Revatio
- Meriana ea ho phekola lefu lena: Latuda, Orap
- Meriana ea kankere: Camptosar, Campto
- Li-derivatives tse nang le anti-migraine tse nang le Ergot: DHE 45, Ergotrate, Hydergine, Migranal
- Meriana e thibelang lefuba ea Rifampin: Mycobutin, Rifater, Rifamate, Rimactane, Rifadin, Priftin
- Litlhaloso: Dormicum, Halcion, Hypam, Hyponvel, Trilam, Versed
- Mokhoakho oa St. John's
Litšebelisano tsa meriana ea mafu a meriana
Tšebeliso ea Prezcobix ka lithethefatsi tse latelang tsa kokoana-hloko e ka fella ka ho lahleheloa ke phekolo ea meriana e tsamaeang le eona kapa kotsi e eketsehileng ea litla-morao:
- Crixivan (indinavir) ha ea lokela ho laoloa ke Prezcobix.
- Videx (didanosine) e lokela ho nkoa ka hora e le 'ngoe pele ho nako e le' ngoe ka mor'a ho nka Prezcobix.
- Intelence (etravirine) ha ea lokela ho laoloa ke Prezcobix.
- Viramune (nevirapine) ha ea lokela ho laoloa ke Prezcobix
- Tekanyo ea Selzentry (maraviroc) e lokela ho fetoloa ho 150mg ka letsatsi le leng le le leng haeba e sebelisoa le Prezcobix.
Litšebelisano tse ling kapa mekhoa e meng
- Tsebisa ngaka ea hao ka boemo leha e le bofe bo tsejoang kapa bo nahanoang hore u na le liphio pele u qala Prezcobix.
- Meriana ea ho se sebetse ea Erectile (Viagra, Levitra, Cialis) e lokela ho sebelisoa ka hloko ha motsoako oa cobicistat oa Prezcobix o ka matlafatsa litla-morao tse bohloko, ho kenyeletsa khathatso ea pono, hypotension, le priapism (e bohloko, e tsitsitseng erections). Ho kgothaletswa hore Viagra tekanyo e fokotsehe ho feta 25mg ka lihora tse 48; Litekanyetso tsa Levitra li fokotsehile ho feta li-2.5mg lihora tse 72, 'me tekanyo ea Cialis e fokotsehile ho fihlela ho feta 10mg ka lihora tse 72.
Lisebelisoa:
Bristol-Myers Squibb. "PREZCOBIX - LINTHO TSA BOHLOKOA TSE BOLETSENG." New York, New York